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Oxatomide

Editor-In-Chief: C. Michael Gibson, M.S., M.D. [1]

Overview

Oxatomide (R35443) is a first-generation antihistamine of the phenylpiperazine class.[1] It was discovered at Janssen Pharmaceutica in 1975. Oxatomide lacks any anticholinergic effects.[1] In addition to its H1 receptor antagonism, it also possesses antiserotonergic actions.[1]

See also

References

  1. 1.0 1.1 1.2 Ohmori K, Ishii H, Nito M, Shuto K, Nakamizo N (May 1983). “[Pharmacological studies on oxatomide (KW-4354). (7) Antagonistic effects on chemical mediators]”. Nippon Yakurigaku Zasshi. Folia Pharmacologica Japonica (in Japanese). 81 (5): 399–409. doi:10.1254/fpj.81.399. PMID 6138301.

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